Endothelin Receptor Inhibitors

ET_A

ET_B

Endothelin Receptor Inhibitors, Agonists, Antagonists & Activators

Product Name	ET_A	ET_B	Purity
Endothelin 1 (swine, human)	ET_A	ET_B	99.12%
Ambrisentan	ET_A		99.95%
Macitentan	ET_A	ET_B	99.87%
BQ-788		ET_B	99.70%
HJP 272	ET_A, IC₅₀: 37.01 nM	ET_B, IC₅₀: 15602.3 nM
Aprocitentan	ET_A, IC₅₀: 3.4 nM ET_A, pA2: 6.7	ET_B, IC₅₀: 987 nM ET_B, pA2: 5.5	99.55%
Sitaxsentan sodium	ET_A, IC₅₀: 1.4 nM ET_A, Ki: 0.43 nM	ET_B, IC₅₀: 9800 nM	98.83%
BQ-123	ET_A		99.91%
BQ-788 sodium salt		ET_B	99.33%
Sulfisoxazole	ET_A, IC₅₀: 0.60 μM	ET_B, IC₅₀: 22 μM	99.90%
Zibotentan	ET_A, Ki: 13 nM		99.37%
IRL-1620 TFA		ET_B	98.73%
Delphinidin 3-rutinoside chloride		ET_B	98.83%
IRL-1620		ET_B	99.69%
Tezosentan	ET_A, pA2: 9.5	ET_B, pA2: 7.7	98.27%
IRL 2500	ET_A, IC₅₀: 94 nM	ET_B, IC₅₀: 1.3 nM	99.27%
A-192621	ET_A, IC₅₀: 4280 nM ET_A, Ki: 5600 nM	ET_B, IC₅₀: 4.5 nM ET_B, Ki: 8.8 nM	99.92%
Schisantherin D		ET_B	99.66%
Avosentan	ET_A		98.15%
Aprocitentan-d₄	ET_A, IC₅₀: 3.4 nM ET_A, pA2: 6.7	ET_B, IC₅₀: 987 nM ET_B, pA2: 5.5	98.76%
Sarafotoxin S6a	ET_A	ET_B	98.45%
BMS 182874	ET_A, IC₅₀: 0.15 μM ET_A, Ki: 0.055 μM		99.85%
Macitentan-d₄	ET_A	ET_B
Ro 46-8443	ET_A, IC₅₀: 6800 nM	ET_B, IC₅₀: 34-69 nM	98.93%
Nebentan	ET_A, Ki: 0.697 nM	ET_B, Ki: 569 nM	99.67%
Nebentan potassium	ET_A, Ki: 0.679 nM	ET_B, Ki: 569 nM	99.53%
J-104132	ET_A, Ki: 0.034 nM	ET_B, Ki: 0.104 nM
[Ala1,3,11,15]-Endothelin (53-63) TFA		ET_B	98.18%
Ro 46-2005	ET_A		98.32%
Edonentan	ET_A, Ki: 10 pM	ET_B, Ki: 810 nM	99.13%
PD-156707	ET_A, Ki: 0.17 μM	ET_B, Ki: 133.8 μM	99.92%
ABT-546	ET_A, Ki: 0.46 nM
Ambrisentan sodium	ET_A
Endothelin 1 (swine, human), Alexa Fluor 488-labeled	ET_A	ET_B
BMS-193884	ET_A, Ki: 1.4 nM	ET_B, Ki: 18700 nM
RES-701-1		ET_B, IC₅₀: 10 nM
SB 247083	ET_A, Ki: 0.41 nM	ET_B, Ki: 467 nM
Sarafotoxin S6a TFA	ET_A	ET_B
Edonentan hydrate	ET_A, Ki: 10 pM
Sulfisoxazole diethanolamine	ET_A, IC₅₀: 0.60 μM	ET_B, IC₅₀: 22 μM
S-1255	ET_A
BMS-187308	ET_A, Ki: 4.7 nM	ET_B, Ki: 1.7 μM
CI-1020	ET_A, IC₅₀: 0.3 nM
BQ-3020		ET_B, IC₅₀: 0.2 nM
PD 155080	ET_A
BQ-610	ET_A
Sitaxsentan	ET_A, IC₅₀: 1.4 nM ET_A, Ki: 0.43 nM	ET_B, IC₅₀: 9800 nM
Sitaxsentan-¹³C₆	ET_A, IC₅₀: 1.4 nM ET_A, Ki: 0.43 nM	ET_B, IC₅₀: 9800 nM
FR139317	ET_A
WS009B	ET_A, IC₅₀: 0.67 μM	ET_B, IC₅₀: 0.8 μM
ATZ-1993	ET_A, pKi: 8.69	ET_B, pKi: 7.20
Sitaxsentan sodium (Standard)	ET_A, IC₅₀: 1.4 nM ET_A, Ki: 0.43 nM	ET_B, IC₅₀: 9800 nM
ZD-1611	ET_A

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